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Tasir Haque
Tasir Haque
Principal Scientist
Verified email at contexttherapeutics.com
Title
Cited by
Cited by
Year
Stereochemical requirements for β-hairpin formation: model studies with four-residue peptides and depsipeptides
TS Haque, JC Little, SH Gellman
Journal of the American Chemical Society 118 (29), 6975-6985, 1996
3181996
Insights on β-hairpin stability in aqueous solution from peptides with enforced type i ‘and type ii ‘β-turns
TS Haque, SH Gellman
Journal of the American Chemical Society 119 (9), 2303-2304, 1997
3061997
Potent, low-molecular-weight non-peptide inhibitors of malarial aspartyl protease plasmepsin II
TS Haque, AG Skillman, CE Lee, H Habashita, IY Gluzman, TJA Ewing, ...
Journal of Medicinal Chemistry 42 (8), 1428-1440, 1999
2231999
Novel uncomplexed and complexed structures of plasmepsin II, an aspartic protease from Plasmodium falciparum
OA Asojo, SV Gulnik, E Afonina, B Yu, JA Ellman, TS Haque, AM Silva
Journal of molecular biology 327 (1), 173-181, 2003
1612003
" Mirror image" reverse turns promote. beta.-hairpin formation
TS Haque, JC Little, SH Gellman
Journal of the American Chemical Society 116 (9), 4105-4106, 1994
1491994
Novel cathepsin D inhibitors block the formation of hyperphosphorylated tau fragments in hippocampus
X Bi, TS Haque, J Zhou, AG Skillman, B Lin, CE Lee, ID Kuntz, JA Ellman, ...
Journal of neurochemistry 74 (4), 1469-1477, 2000
992000
Parallel Synthesis of Potent, Pyrazole-Based Inhibitors of Helicobacter p ylori Dihydroorotate Dehydrogenase
TS Haque, S Tadesse, J Marcinkeviciene, MJ Rogers, C Sizemore, ...
Journal of medicinal chemistry 45 (21), 4669-4678, 2002
922002
Searching for minimum increments of hydrophobic collapse: flexible dinaphthyl carboxylates
LF Newcomb, TS Haque, SH Gellman
Journal of the American Chemical Society 117 (24), 6509-6519, 1995
841995
Helicobacter pylori-selective antibacterials based on inhibition of pyrimidine biosynthesis
RA Copeland, J Marcinkeviciene, TS Haque, LM Kopcho, W Jiang, ...
Journal of Biological Chemistry 275 (43), 33373-33378, 2000
702000
Selective inhibition of bacterial dihydroorotate dehydrogenases by thiadiazolidinediones
J Marcinkeviciene, MJ Rogers, L Kopcho, W Jiang, K Wang, DJ Murphy, ...
Biochemical pharmacology 60 (3), 339-342, 2000
652000
Optimizing preparative LC/MS configurations and methods for parallel synthesis purification
KF Blom, R Sparks, J Doughty, JG Everlof, T Haque, AP Combs
Journal of Combinatorial Chemistry 5 (5), 670-683, 2003
512003
Structural Characterization of Thiocyclophanes That Promote Edge-to-Face Aromatic-Aromatic Geometries
KD Schladetzky, TS Haque, SH Gellman
The Journal of Organic Chemistry 60 (13), 4108-4113, 1995
511995
New evidence that the hydrophobic effect and dispersion are not major driving forces for nucleotide base stacking.
SH Gellman, TS Haque, LF Newcomb
Biophysical journal 71 (6), 3523, 1996
491996
N-Arylation of primary and secondary aliphatic amines on solid supports
AP Combs, S Tadesse, M Rafalski, TS Haque, PYS Lam
Journal of Combinatorial Chemistry 4 (2), 179-182, 2002
472002
Human glucagon-like-peptide-1 modulators and their use in treatment of diabetes and related conditions
WR Ewing, C Mapelli, RB Sulsky, TS Haque, VG Lee, DJ Riexinger, ...
US Patent 7,417,028, 2008
402008
Identification of potent 11mer glucagon-like peptide-1 receptor agonist peptides with novel C-terminal amino acids: homohomophenylalanine analogs
TS Haque, VG Lee, D Riexinger, M Lei, S Malmstrom, L Xin, S Han, ...
Peptides 31 (5), 950-955, 2010
262010
Pyrazolobenzamides and derivatives as factor Xa inhibitors
PY Lam, CG Clark, R Li, TS Haque, KA Rossi
US Patent 7,381,732, 2008
262008
Potent biphenyl-and 3-phenyl pyridine-based inhibitors of acetyl-CoA carboxylase
TS Haque, N Liang, R Golla, R Seethala, Z Ma, WR Ewing, CB Cooper, ...
Bioorganic & medicinal chemistry letters 19 (20), 5872-5876, 2009
242009
Differential activation of recombinant human acetyl-CoA carboxylases 1 and 2 by citrate
GA Locke, D Cheng, MR Witmer, JK Tamura, T Haque, RF Carney, ...
Archives of biochemistry and biophysics 475 (1), 72-79, 2008
242008
Liquid-liquid extraction coupled with LC/MS/MS for monitoring of malonyl-CoA in rat brain tissue
JM Onorato, L Chen, P Shipkova, Z Ma, AV Azzara, JJ Devenny, N Liang, ...
Analytical and bioanalytical chemistry 397, 3137-3142, 2010
222010
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