| Design of remarkably simple, yet potent urea-based inhibitors of glutamate carboxypeptidase II (NAALADase) AP Kozikowski, F Nan, P Conti, J Zhang, E Ramadan, T Bzdega, ... Journal of medicinal chemistry 44 (3), 298-301, 2001 | 338 | 2001 |
| Synthesis and Biochemical Evaluation of Δ2-Isoxazoline Derivatives as DNA Methyltransferase 1 Inhibitors S Castellano, D Kuck, M Viviano, J Yoo, F López-Vallejo, P Conti, ... Journal of medicinal chemistry 54 (21), 7663-7677, 2011 | 193 | 2011 |
| Synthesis of new Δ2-isoxazoline derivatives and their pharmacological characterization as β-adrenergic receptor antagonists P Conti, C Dallanoce, M De Amici, C De Micheli, KN Klotz Bioorganic & medicinal chemistry 6 (4), 401-408, 1998 | 129 | 1998 |
| Drug discovery targeting amino acid racemases P Conti, L Tamborini, A Pinto, A Blondel, P Minoprio, A Mozzarelli, ... Chemical reviews 111 (11), 6919-6946, 2011 | 125 | 2011 |
| Inhibition of rhodesain as a novel therapeutic modality for human African trypanosomiasis R Ettari, L Tamborini, IC Angelo, N Micale, A Pinto, C De Micheli, P Conti Journal of Medicinal Chemistry 56 (14), 5637-5658, 2013 | 99 | 2013 |
| A regioselective route to 5-substituted pyrazole-and pyrazoline-3-phosphonic acids and esters P Conti, A Pinto, L Tamborini, V Rizzo, C De Micheli Tetrahedron 63 (25), 5554-5560, 2007 | 88 | 2007 |
| The glial glutamate transporter 1 (GLT1) is expressed by pancreatic β-cells and prevents glutamate-induced β-cell death ES Di Cairano, AM Davalli, L Perego, S Sala, VF Sacchi, S La Rosa, ... Journal of Biological Chemistry 286 (16), 14007-14018, 2011 | 79 | 2011 |
| An efficient method for the lipase-catalysed resolution and in-line purification of racemic flurbiprofen in a continuous-flow reactor L Tamborini, D Romano, A Pinto, A Bertolani, F Molinari, P Conti Journal of Molecular Catalysis B: Enzymatic 84, 78-82, 2012 | 60 | 2012 |
| UCP2 inhibition induces ROS/Akt/mTOR axis: Role of GAPDH nuclear translocation in genipin/everolimus anticancer synergism I Dando, R Pacchiana, E Dalla Pozza, I Cataldo, S Bruno, P Conti, ... Free Radical Biology and Medicine 113, 176-189, 2017 | 59 | 2017 |
| Synthesis and functional characterization of novel derivatives related to oxotremorine and oxotremorine-M C Dallanoce, P Conti, M De Amici, C De Micheli, E Barocelli, M Chiavarini, ... Bioorganic & medicinal chemistry 7 (8), 1539-1547, 1999 | 58 | 1999 |
| Discovery of covalent inhibitors of glyceraldehyde-3-phosphate dehydrogenase, a target for the treatment of malaria S Bruno, A Pinto, G Paredi, L Tamborini, C De Micheli, V La Pietra, ... Journal of Medicinal Chemistry 57 (17), 7465-7471, 2014 | 57 | 2014 |
| Synthesis, binding affinity at glutamic acid receptors, neuroprotective effects, and molecular modeling investigation of novel dihydroisoxazole amino acids P Conti, M De Amici, G Grazioso, G Roda, A Pinto, KB Hansen, B Nielsen, ... Journal of medicinal chemistry 48 (20), 6315-6325, 2005 | 57 | 2005 |
| An efficient continuous flow process for the synthesis of a non-conventional mixture of fructooligosaccharides P Zambelli, L Tamborini, S Cazzamalli, A Pinto, S Arioli, S Balzaretti, ... Food Chemistry 190, 607-613, 2016 | 53 | 2016 |
| Mutant p53 prevents GAPDH nuclear translocation in pancreatic cancer cells favoring glycolysis and 2-deoxyglucose sensitivity G Butera, R Pacchiana, N Mullappilly, M Margiotta, S Bruno, P Conti, ... Biochimica et Biophysica Acta (BBA)-Molecular Cell Research 1865 (12), 1914-1923, 2018 | 50 | 2018 |
| Chemoenzymatic synthesis in flow reactors: A rapid and convenient preparation of Captopril V De Vitis, F Dall'Oglio, A Pinto, C De Micheli, F Molinari, P Conti, ... ChemistryOpen 6 (5), 668-673, 2017 | 50 | 2017 |
| Flow-based stereoselective reduction of ketones using an immobilized ketoreductase/glucose dehydrogenase mixed bed system F Dall'Oglio, ML Contente, P Conti, F Molinari, D Monfredi, A Pinto, ... Catalysis Communications 93, 29-32, 2017 | 50 | 2017 |
| Design and synthesis of novel isoxazole-based HDAC inhibitors P Conti, L Tamborini, A Pinto, L Sola, R Ettari, C Mercurio, C De Micheli European journal of medicinal chemistry 45 (9), 4331-4338, 2010 | 50 | 2010 |
| Synthesis and enantiopharmacology of new AMPA-kainate receptor agonists P Conti, M De Amici, G De Sarro, M Rizzo, TB Stensbøl, ... Journal of medicinal chemistry 42 (20), 4099-4107, 1999 | 48 | 1999 |
| Development of rhodesain inhibitors with a 3‐bromoisoxazoline warhead R Ettari, L Tamborini, IC Angelo, S Grasso, T Schirmeister, L Lo Presti, ... ChemMedChem 8 (12), 2070-2076, 2013 | 46 | 2013 |
| Biotransformation with whole microbial systems in a continuous flow reactor: resolution of (RS)-flurbiprofen using Aspergillus oryzae by direct esterification with ethanol in … L Tamborini, D Romano, A Pinto, M Contente, MC Iannuzzi, P Conti, ... Tetrahedron letters 54 (45), 6090-6093, 2013 | 43 | 2013 |
