| Selective inhibition of factor inhibiting hypoxia-inducible factor MA McDonough, LA McNeill, M Tilliet, CA Papamicaël, QY Chen, ... Journal of the American Chemical Society 127 (21), 7680-7681, 2005 | 165 | 2005 |
| The 1.5-Å structure of Chryseobacterium meningosepticum zinc β-lactamase in complex with the inhibitor, D-captopril I García-Sáez, J Hopkins, C Papamicaël, N Franceschini, G Amicosante, ... Journal of biological chemistry 278 (26), 23868-23873, 2003 | 161 | 2003 |
| Thiomandelic Acid, a Broad Spectrum Inhibitor of Zinc β-Lactamases: KINETIC AND SPECTROSCOPIC STUDIES* 210 C Mollard, C Moali, C Papamicael, C Damblon, S Vessilier, G Amicosante, ... Journal of Biological Chemistry 276 (48), 45015-45023, 2001 | 159 | 2001 |
| Three-dimensional structure of FEZ-1, a monomeric subclass B3 metallo-β-lactamase from Fluoribacter gormanii, in native form and in complex with D-captopril I Garcıa-Sáez, PS Mercuri, C Papamicaël, R Kahn, JM Frère, M Galleni, ... Journal of molecular biology 325 (4), 651-660, 2003 | 157 | 2003 |
| Structural basis for the broad-spectrum inhibition of metallo-β-lactamases by thiols BMR Liénard, G Garau, L Horsfall, AI Karsisiotis, C Damblon, P Lassaux, ... Organic & biomolecular chemistry 6 (13), 2282-2294, 2008 | 153 | 2008 |
| Modular synthesis of benzene-centered porphyrin trimers and a dendritic porphyrin hexamer O Mongin, C Papamicaël, N Hoyler, A Gossauer The Journal of Organic Chemistry 63 (16), 5568-5580, 1998 | 135 | 1998 |
| Coordination geometries of metal ions in D-or L-captopril-inhibited metallo-β-lactamases U Heinz, R Bauer, S Wommer, W Meyer-Klaucke, C Papamichaels, ... Journal of Biological Chemistry 278 (23), 20659-20666, 2003 | 107 | 2003 |
| Investigations of electronic energy transfer dynamics in multiporphyrin arrays P Brodard, S Matzinger, E Vauthey, O Mongin, C Papamicaël, A Gossauer The Journal of Physical Chemistry A 103 (30), 5858-5870, 1999 | 97 | 1999 |
| Donepezil-based central acetylcholinesterase inhibitors by means of a “bio-oxidizable” prodrug strategy: design, synthesis, and in vitro biological evaluation L Peauger, R Azzouz, V Gembus, ML Tintas, ... Journal of medicinal chemistry 60 (13), 5909-5926, 2017 | 80 | 2017 |
| The inhibitor thiomandelic acid binds to both metal ions in metallo-β-lactamase and induces positive cooperativity in metal binding C Damblon, M Jensen, A Ababou, I Barsukov, C Papamicael, ... Journal of Biological Chemistry 278 (31), 29240-29251, 2003 | 60 | 2003 |
| ortho-Lithiation of S-tert-butyl-S-phenylsulfoximines. New route to enantiopure sulfinamides via a de-tert-butylation reaction S Gaillard, C Papamicaël, G Dupas, F Marsais, V Levacher Tetrahedron 61 (34), 8138-8147, 2005 | 54 | 2005 |
| An overview of the synthesis of highly versatile N-hydroxysuccinimide esters A Barre, ML Ţînţaş, V Levacher, C Papamicaël, V Gembus Synthesis 49 (03), 472-483, 2017 | 47 | 2017 |
| Novel donepezil-like N-benzylpyridinium salt derivatives as AChE inhibitors and their corresponding dihydropyridine “bio-oxidizable” prodrugs: Synthesis, biological evaluation … R Azzouz, L Peauger, V Gembus, ML Ţînţaş, ... European journal of medicinal chemistry 145, 165-190, 2018 | 36 | 2018 |
| New development of Meyers’ methodology: stereoselective preparation of an axially chiral 5, 7-fused bicyclic lactam related to circumdatins/benzomalvins and asperlicins M Penhoat, P Bohn, G Dupas, C Papamicaël, F Marsais, V Levacher Tetrahedron: Asymmetry 17 (2), 281-286, 2006 | 35 | 2006 |
| Preparation of new axially chiral bridged 2, 2′-bipyridines and pyridyl monooxazolines (pymox). Evaluation in copper (i)-catalyzed enantioselective cyclopropanation A Bouet, B Heller, C Papamicaël, G Dupas, S Oudeyer, F Marsais, ... Organic & Biomolecular Chemistry 5 (9), 1397-1404, 2007 | 33 | 2007 |
| Rational design of central selective acetylcholinesterase inhibitors by means of a “bio-oxidisable prodrug” strategy P Bohn, N Le Fur, G Hagues, J Costentin, N Torquet, C Papamicaël, ... Organic & biomolecular chemistry 7 (12), 2612-2618, 2009 | 32 | 2009 |
| Palladium-Catalyzed Carbonylation of (Hetero)Aryl, Alkenyl and Allyl Halides by Means of N-Hydroxysuccinimidyl Formate as CO Surrogate A Barré, ML Tintas, F Alix, V Gembus, C Papamicael, V Levacher The Journal of Organic Chemistry 80 (13), 6537-6544, 2015 | 30 | 2015 |
| Meyers’ bicyclic lactam formation under mild and highly stereoselective conditions M Penhoat, S Leleu, G Dupas, C Papamicaël, F Marsais, V Levacher Tetrahedron letters 46 (48), 8385-8389, 2005 | 29 | 2005 |
| Preparation of axially chiral quinolinium salts related to NAD+ models: new investigations of these biomimetic models as ‘chiral amide-transferring agents’ S Leleu, C Papamicaël, F Marsais, G Dupas, V Levacher Tetrahedron: Asymmetry 15 (24), 3919-3928, 2004 | 29 | 2004 |
| Amine capture strategy for peptide bond formation by means of quinolinium thioester salts S Leleu, M Penhoat, A Bouet, G Dupas, C Papamicaël, F Marsais, ... Journal of the American Chemical Society 127 (45), 15668-15669, 2005 | 28 | 2005 |
Stéphane LELEUDoctorVerified email at univ-rouen.fr
