3,4-Dihydropyrimidin-2(1H)-ones as Antagonists of the Human A2B Adenosine Receptor: Optimization, Structure–Activity Relationship Studies, and … M Majellaro, W Jespers, A Crespo, MJ Núñez, S Novio, J Azuaje, ... Journal of Medicinal Chemistry 64 (1), 458-480, 2020 | 24 | 2020 |
Nitrogen-Walk Approach to Explore Bioisosteric Replacements in a Series of Potent A2B Adenosine Receptor Antagonists A Mallo-Abreu, R Prieto-Díaz, W Jespers, J Azuaje, M Majellaro, ... Journal of Medicinal Chemistry 63 (14), 7721-7739, 2020 | 23 | 2020 |
Trifluorinated Pyrimidine-Based A2B Antagonists: Optimization and Evidence of Stereospecific Recognition A Mallo-Abreu, M Majellaro, W Jespers, J Azuaje, O Caamano, ... Journal of Medicinal Chemistry 62 (20), 9315-9330, 2019 | 18 | 2019 |
Catalytic performance of a metal-free graphene oxide-Al2O3 composite assembled by 3D printing J Azuaje, A Rama, A Mallo-Abreu, MG Boado, M Majellaro, CR Tubío, ... Journal of the European Ceramic Society 41 (2), 1399-1406, 2021 | 14 | 2021 |
Exploring the Effect of Halogenation in a Series of Potent and Selective A2B Adenosine Receptor Antagonists R Prieto-Díaz, M González-Gómez, H Fojo-Carballo, J Azuaje, ... Journal of Medicinal Chemistry 66 (1), 890-912, 2022 | 9 | 2022 |
Exploring Non-orthosteric Interactions with a Series of Potent and Selective A3 Antagonists D Miranda-Pastoriza, R Bernárdez, J Azuaje, R Prieto-Díaz, M Majellaro, ... ACS Medicinal Chemistry Letters 13 (2), 243-249, 2022 | 5 | 2022 |
Potent and Subtype-Selective Dopamine D2 Receptor Biased Partial Agonists Discovered via an Ugi-Based Approach A Mallo-Abreu, I Reyes-Resina, J Azuaje, R Franco, A García-Rey, ... Journal of Medicinal Chemistry 64 (12), 8710-8726, 2021 | 4 | 2021 |
Exploring Biginelli-based scaffolds as A2B adenosine receptor antagonists: Unveiling novel structure-activity relationship trends, lead compounds, and potent colorectal … R Prieto-Díaz, H Fojo-Carballo, M Majellaro, T Tandarić, J Azuaje, J Brea, ... Biomedicine & pharmacotherapy 173, 116345, 2024 | | 2024 |
New ligands and pharmacological tools for the study of g protein-coupled receptors using multicomponent reactions AM Abreu New ligands and pharmacological tools for the study of g protein-coupled …, 2021 | | 2021 |
3, 4-Dihydropyrimidin-2 (1H)-ones as Antagonists of the Human A2B Adenosine Receptor: Optimization, Structure–Activity Relationship Studies, and Enantiospecific Recognition M Majellaro, W Jespers, A Crespo, MJ Núñez, S Novio, J Azuaje, ... Journal of Medicinal Chemistry 64 (1), 458-480, 2021 | | 2021 |
Exploring the Effect of Halogenation in a Series of Potent and Selective A2B Adenosine Receptor Antagonists MR Paleo Pillado, R Prieto Díaz, M González Gómez, H Fojo Carballo, ... ACS Publications, 0 | | |
New Ligands and Pharmacological Tools for the Study of G Protein-Coupled Receptors Using Multicomponent Reactions A Mallo Abreu | | |
A Nitrogen-Walk Approach to Explore Bioisosteric Replacements in a Series of Potent A2B Adenosine Receptor Antagonists MA Ana, PD Ruben, J Willem, A Jhonny, M Maria, V Carmen, GM Xerardo, ... Journal of medicinal chemistry, 0 | | |